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Sleeping pill found to reduce levels of Alzheimer's proteins (Suvorexant)
Medical Xpress / Washington University School of Medicine / Annals of Neurology ^ | April 20, 2023 | Brendan P. Lucey et al

Posted on 04/22/2023 8:44:41 PM PDT by ConservativeMind

Sleep disturbances can be an early sign of Alzheimer's. It's a vicious cycle: Alzheimer's disease involves changes to the brain that disrupt sleep, and poor sleep accelerates harmful changes to the brain.

Researchers have identified a possible way to help break that cycle. A small, two-night study has shown that people who took a sleeping pill before bed experienced a drop in the levels of key Alzheimer's proteins.

The study involved a sleeping aid known as suvorexant.

Suvorexant belongs to a class of insomnia medications known as dual orexin receptor antagonists. Orexin is a natural biomolecule that promotes wakefulness. When orexin is blocked, people fall asleep.

Alzheimer's disease begins when plaques of the protein amyloid beta start building up in the brain. After years of amyloid accumulation, a second brain protein, tau, begins to form tangles that are toxic to neurons.

The participants were given a lower dose (10 mg) of suvorexant (13 people), a higher dose (20 mg) of suvorexant (12 people) or a placebo (13 people) at 9 p.m. and then went to sleep. Researchers withdrew a small amount of cerebrospinal fluid via spinal tap every two hours for 36 hours, starting one hour before the sleeping aid or placebo was administered, to measure how amyloid and tau levels changed over the next day and a half.

Amyloid levels dropped 10% to 20% in the cerebrospinal fluid of people who had received the high dose of suvorexant compared to people who had received placebo, and the levels of a key form of tau known as hyperphosphorylated tau dropped 10% to 15%, compared to people who had received placebo. Both differences are statistically significant.

A second dose of suvorexant, administered on the second night, sent the levels of both proteins down again for people in the high-dose group.

(Excerpt) Read more at medicalxpress.com ...


TOPICS: Health/Medicine
KEYWORDS: alzheimers; insomnia; sleepingpill
This approach could really extend the time of onset of Alzheimer’s, it would appear.

The drug is currently available.

1 posted on 04/22/2023 8:44:41 PM PDT by ConservativeMind
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To: ConservativeMind

Is it OTC?

CA....


2 posted on 04/22/2023 10:51:45 PM PDT by Chances Are (Seems I've found that silly grin again....)
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To: ConservativeMind

Bring back Quaaludes!

Aside from this they are instant cure for waning female virility

No question of that


3 posted on 04/22/2023 11:10:47 PM PDT by wardaddy (Truth is treason in the Empire of lies)
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BM


4 posted on 04/23/2023 12:45:07 AM PDT by misanthrope (Deranged, sinister, deplorable troll)
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To: ConservativeMind

this was a two night study.


5 posted on 04/23/2023 5:37:26 AM PDT by ckilmer (q)
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To: ConservativeMind

This reads like I would expect, that suvorexant is not itself effective against Alzheimer’s. It suppresses orexin, the body’s wakefulness hormone. Suppressing orexin makes patients sleep, and sleep suppresses inflammation. Inflammation reduction reduces amyloid beta production, and suppresses the onset of Alzheimer’s.

Sleep is key.


6 posted on 04/23/2023 7:09:15 AM PDT by nagant
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